Reviewed by Peptide Treatments Medical Advisory Board (Medical Advisory Board)

Melanotan II: Side Effects & Safety

Known side effects, safety considerations, and adverse reaction data for Melanotan II.

Back to Melanotan II overview

Data source: Side effect data comes from clinical trials, preclinical research, and anecdotal reports. No FDA-approved labeling exists for this compound.

Reported Side Effects (8 items)

# Side Effect
1 MELANOMA — documented case reports at injection sites
2 Nausea — common, dose-related
3 Facial flushing
4 Spontaneous erections / priapism risk (males)
5 Generalized skin darkening
6 Yawning
7 Appetite suppression
8 Systemic toxicity and rhabdomyolysis (case report)

Known Drug Interactions

Important: Only documented and contraindicated interactions are shown here. View all interactions including theoretical →
Drug Classification Mechanism
PDE5 inhibitors (sildenafil, tadalafil) Documented Additive vasodilation and erectile effects — increased risk of hypotension