Reviewed by Peptide Treatments Medical Advisory Board (Medical Advisory Board)

5-Amino-1MQ: Research & Evidence

Early-Stage Research

Published research, clinical trial data, and evidence grading for 5-Amino-1MQ across studied indications.

Back to 5-Amino-1MQ overview

Research Summary

5-Amino-1MQ has zero human studies — it exists entirely in preclinical research. Mouse studies show NNMT inhibition reduces weight gain and improves metabolic markers, but no human pharmacokinetic, safety, or efficacy data exists. Classified as a small molecule quinolinium compound rather than a classical peptide.

Evidence by Indication (2 indications)

Indication Tier Trials Summary
Fat metabolism / obesity Tier D 0 NNMT inhibition reduces fat mass in mouse models; zero human data
NNMT inhibition Tier D 0 Mechanism well-characterized in vitro; no human clinical data exists

Graded using our evidence tier methodology.

Citations (2 sources)

  1. 1. Nicotinamide N-methyltransferase inhibition mitigates obesity-related metabolic dysfunction. Study

    (2024), Diabetes, obesity & metabolism

  2. 2. Reduced calorie diet combined with NNMT inhibition establishes a distinct microbiome in DIO mice. Study

    Dimet-Wiley A, Wu Q, Wiley JT, et al. (2022), Scientific reports